olm, T.N. Tozer. Clinical pharmacokinetics and pharmacodynamics: concepts and applications. Wolters Kluwer Health/Lippincott William & Wilkins, 2011. ISBN 978-0781750097
[2] M. Gibaldi, D. Perrie. Pharmacokinetics 2nd ed. Marcel Dekker, New York, 1982. https://doi.org/10.1201/b14095 DOI: https://doi.org/10.1201/b14095
[3] P. Poulin, F.P. Theil. Prediction of pharmacokinetics prior to in vivo studies. II. Generic physiologically based pharmacokinetic models of drug disposition. Journal of Pharmaceutical Sciences 91(5) (2002) 1358-1370. https://doi.org/10.1002/jps.10128 DOI: https://doi.org/10.1002/jps.10128
[4] A. Rane, G.R. Wilkinson, D.G. Shand. Prediction of hepatic extraction ratio from in vitro measurement of intrinsic clearance. Journal of Pharmacology and Experimental Therapeutics 200(2) (1977) 420-424. https://pubmed.ncbi.nlm.nih.gov/839445/ DOI: https://doi.org/10.1016/S0022-3565(25)30786-X
[5] D. A. Smith, L. Di, E.H. Kerns. The free drug hypothesis: key concepts in drug discovery. Nature Reviews Drug Discovery 9 (2010) 929-939. https://doi.org/10.1038/nrd3287 DOI: https://doi.org/10.1038/nrd3287
[6] Goodman & Gilman's: The Pharmacological Basis of Therapeutics, 14th Edition. L.L. Brunton, B.C. Knollmann, Eds., McGraw-Hill Education; 2023. https://accessmedicine.mhmedical.com/content.aspx?bookid=3191§ionid=265824603
[7] K. Valko. Application of biomimetic HPLC to estimate in vivo behavior of early drug discovery compounds. Future Drug Discovery 1(1) (2019). https://doi.org/10.4155/fdd-2019-0004 DOI: https://doi.org/10.4155/fdd-2019-0004
[8] K.L. Valko. Biomimetic chromatography-A novel application of the chromatographic principles. Analytical Science Advances 3 (2022) 146-153. https://doi.org/10.1002/ansa.202200004 DOI: https://doi.org/10.1002/ansa.202200004
[9] K.L. Valkó, S.B. Nunhuck, A.P. Hill. Estimating Unbound Volume of Distribution and Tissue Binding by in vitro HPLC-based Human Serum Albumin and Immobilized Artificial Membrane-Binding Measurements. Journal of Pharmaceutical Sciences 100 (2011) 849-862. https://doi.org/10.1002/jps.22323 DOI: https://doi.org/10.1002/jps.22323
[10] F. Hollosy, K. Valko, A. Hersey, S. Nunhuck, G. Keri, C. Bevan. Estimation of Volume of Distribution in Humans from HPLC Measurements of Human Serum Albumin Binding and Immobilized Artificial Membrane Partitioning. Journal of Medicinal Chemistry 49 (2006) 6958-6971. https://doi.org/10.1021/jm050957i DOI: https://doi.org/10.1021/jm050957i
[11] K. Valko, E. Chiarparin, S. Nunhuck, D. Montanari. In vitro measurement of drug efficiency index to aid early lead optimization. Journal of Pharmaceutical Sciences 101 (2012) 4155-4169. https://doi.org/10.1002/jps.23305 DOI: https://doi.org/10.1002/jps.23305
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